JJKK 048, Potent and selective MAGL inhibitor, Each
$ 473.28
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Details
JJKK 048 is a potent and selective monoacylglycerol lipase (MAGL) inhibitor (IC50 = 0.4 nM). Exhibits >13,000 and ∽630-fold selectivity for MAGL over FAAH and ABHD6, respectively. Increases brain levels of 2-arachidonoylglycerol (2-AG) levels in mice in vivo. Promotes analgesia in pain models.
Additional Information
SKU | 10514402 |
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UOM | Each |
UNSPSC | 41116105 |
Manufacturer Part Number | 5206/10 |